Discovery of N-(piperidin-3-yl)-N-(pyridin-2-yl)piperidine/piperazine-1-carboxamides as small molecule inhibitors of PCSK9

Publication

Citation
Londregan A., Aspnes G., Limberakis C., Loria P., McClure K., Petersen D., Raymer B., Ruggeri R., Wei L., Xiao J., Piotrowski D.: Discovery of N-(piperidin-3-yl)-N-(pyridin-2-yl)piperidine/piperazine-1-carboxamides as small molecule inhibitors of PCSK9. Bioorganic & Medicinal Chemistry Letters, Volume 28 (23-24), 2018
Authors
Allyn T. Londregan, Gary Aspnes, Chris Limberakis, Paula M. Loria, Kim F. McClure, Donna N. Petersen, Brian Raymer, Roger B. Ruggeri, Liuqing Wei, Jun Xiao, David W. Piotrowski
Journal
Bioorganic & Medicinal Chemistry Letters
Year
2018
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Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

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