{"data":{"id":4794,"citation":"Londregan A., Aspnes G., Limberakis C., Loria P., McClure K., Petersen D., Raymer B., Ruggeri R., Wei L., Xiao J., Piotrowski D.: Discovery of N-(piperidin-3-yl)-N-(pyridin-2-yl)piperidine\/piperazine-1-carboxamides as small molecule inhibitors of PCSK9. Bioorganic &amp; Medicinal Chemistry Letters, Volume 28 (23-24), 2018","title":"Discovery of N-(piperidin-3-yl)-N-(pyridin-2-yl)piperidine\/piperazine-1-carboxamides as small molecule inhibitors of PCSK9","doi":"10.1016\/j.bmcl.2018.10.029","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2018.10.029","pmid":null,"year":2018,"journal":"Bioorganic &amp; Medicinal Chemistry Letters","volume":"28","issue":"23-24","page":null,"authors":[{"first_name":"Allyn T.","last_name":"Londregan","full_name":"Allyn T. Londregan"},{"first_name":"Gary","last_name":"Aspnes","full_name":"Gary Aspnes"},{"first_name":"Chris","last_name":"Limberakis","full_name":"Chris Limberakis"},{"first_name":"Paula M.","last_name":"Loria","full_name":"Paula M. Loria"},{"first_name":"Kim F.","last_name":"McClure","full_name":"Kim F. McClure"},{"first_name":"Donna N.","last_name":"Petersen","full_name":"Donna N. Petersen"},{"first_name":"Brian","last_name":"Raymer","full_name":"Brian Raymer"},{"first_name":"Roger B.","last_name":"Ruggeri","full_name":"Roger B. Ruggeri"},{"first_name":"Liuqing","last_name":"Wei","full_name":"Liuqing Wei"},{"first_name":"Jun","last_name":"Xiao","full_name":"Jun Xiao"},{"first_name":"David W.","last_name":"Piotrowski","full_name":"David W. Piotrowski"}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/4794","landing_page":"https:\/\/molmedb.upol.cz\/publication\/4794","created_at":"2026-06-22T14:33:15.000000Z","updated_at":"2026-06-22T14:33:15.000000Z"}}