Discovery of Dihydrobenzoxazepinone (GS-6615) Late Sodium Current Inhibitor (Late I<sub>Na</sub>i), a Phase II Agent with Demonstrated Preclinical Anti-Ischemic and Antiarrhythmic Properties.

Publication

Citation
Zablocki JA, Elzein E, Li X, Koltun DO, Parkhill EQ, Kobayashi T, Martinez R, Corkey B, Jiang H, Perry T, Kalla R, Notte GT, Saunders O, Graupe M, Lu Y, Venkataramani C, Guerrero J, Perry J, Osier M, Strickley R, Liu G, Wang WQ, Hu L, Li XJ, El-Bizri N, Hirakawa R, Kahlig K, Xie C, Li CH, Dhalla AK, Rajamani S, Mollova N, Soohoo D, Lepist EI, Murray B, Rhodes G, Belardinelli L, Desai MC.: Discovery of Dihydrobenzoxazepinone (GS-6615) Late Sodium Current Inhibitor (Late I<sub>Na</sub>i), a Phase II Agent with Demonstrated Preclinical Anti-Ischemic and Antiarrhythmic Properties. J Med Chem, Volume 59 (19), 2016
Authors
Belardinelli L, Corkey B, Desai MC., Dhalla AK, El-Bizri N, Elzein E, Graupe M, Guerrero J, Hirakawa R, Hu L, Jiang H, Kahlig K, Kalla R, Kobayashi T, Koltun DO, Lepist EI, Li CH, Li X, Li XJ, Liu G, Lu Y, Martinez R, Mollova N, Murray B, Notte GT, Osier M, Parkhill EQ, Perry J, Perry T, Rajamani S, Rhodes G, Saunders O, Soohoo D, Strickley R, Venkataramani C, Wang WQ, Xie C, Zablocki JA
Journal
J Med Chem
Year
2016
PubMed
27690427
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Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

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