{"data":{"id":4046,"citation":"Zablocki JA, Elzein E, Li X, Koltun DO, Parkhill EQ, Kobayashi T, Martinez R, Corkey B, Jiang H, Perry T, Kalla R, Notte GT, Saunders O, Graupe M, Lu Y, Venkataramani C, Guerrero J, Perry J, Osier M, Strickley R, Liu G, Wang WQ, Hu L, Li XJ, El-Bizri N, Hirakawa R, Kahlig K, Xie C, Li CH, Dhalla AK, Rajamani S, Mollova N, Soohoo D, Lepist EI, Murray B, Rhodes G, Belardinelli L, Desai MC.: Discovery of Dihydrobenzoxazepinone (GS-6615) Late Sodium Current Inhibitor (Late I<sub>Na<\/sub>i), a Phase II Agent with Demonstrated Preclinical Anti-Ischemic and Antiarrhythmic Properties. J Med Chem, Volume 59 (19), 2016","title":"Discovery of Dihydrobenzoxazepinone (GS-6615) Late Sodium Current Inhibitor (Late I<sub>Na<\/sub>i), a Phase II Agent with Demonstrated Preclinical Anti-Ischemic and Antiarrhythmic Properties.","doi":"10.1021\/acs.jmedchem.6b00939","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.6b00939","pmid":"27690427","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/27690427\/","year":2016,"journal":"J Med Chem","volume":"59","issue":"19","page":"9005-9017","authors":[{"first_name":"Belardinelli L","last_name":null,"full_name":null},{"first_name":"Corkey B","last_name":null,"full_name":null},{"first_name":"Desai MC.","last_name":null,"full_name":null},{"first_name":"Dhalla AK","last_name":null,"full_name":null},{"first_name":"El-Bizri N","last_name":null,"full_name":null},{"first_name":"Elzein E","last_name":null,"full_name":null},{"first_name":"Graupe M","last_name":null,"full_name":null},{"first_name":"Guerrero J","last_name":null,"full_name":null},{"first_name":"Hirakawa R","last_name":null,"full_name":null},{"first_name":"Hu L","last_name":null,"full_name":null},{"first_name":"Jiang H","last_name":null,"full_name":null},{"first_name":"Kahlig K","last_name":null,"full_name":null},{"first_name":"Kalla R","last_name":null,"full_name":null},{"first_name":"Kobayashi T","last_name":null,"full_name":null},{"first_name":"Koltun DO","last_name":null,"full_name":null},{"first_name":"Lepist EI","last_name":null,"full_name":null},{"first_name":"Li CH","last_name":null,"full_name":null},{"first_name":"Li X","last_name":null,"full_name":null},{"first_name":"Li XJ","last_name":null,"full_name":null},{"first_name":"Liu G","last_name":null,"full_name":null},{"first_name":"Lu Y","last_name":null,"full_name":null},{"first_name":"Martinez R","last_name":null,"full_name":null},{"first_name":"Mollova N","last_name":null,"full_name":null},{"first_name":"Murray B","last_name":null,"full_name":null},{"first_name":"Notte GT","last_name":null,"full_name":null},{"first_name":"Osier M","last_name":null,"full_name":null},{"first_name":"Parkhill EQ","last_name":null,"full_name":null},{"first_name":"Perry J","last_name":null,"full_name":null},{"first_name":"Perry T","last_name":null,"full_name":null},{"first_name":"Rajamani S","last_name":null,"full_name":null},{"first_name":"Rhodes G","last_name":null,"full_name":null},{"first_name":"Saunders O","last_name":null,"full_name":null},{"first_name":"Soohoo D","last_name":null,"full_name":null},{"first_name":"Strickley R","last_name":null,"full_name":null},{"first_name":"Venkataramani C","last_name":null,"full_name":null},{"first_name":"Wang WQ","last_name":null,"full_name":null},{"first_name":"Xie C","last_name":null,"full_name":null},{"first_name":"Zablocki JA","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/4046","landing_page":"https:\/\/molmedb.upol.cz\/publication\/4046","created_at":"2024-05-21T20:14:48.000000Z","updated_at":null}}