Preparation and optimization of new 4-(2-(indolin-1-yl)-2-oxoethyl)-2-morpholinothiazole-5-carboxylic acid and amide derivatives as potent and selective PI3Kβ inhibitors.

Citation: Certal V, Halley F, Virone-Oddos A, Filoche-Rommé B, Carry JC, Gruss-Leleu F, Bertin L, Guizani H, Pilorge F, Richepin P, Karlsson A, Charrier V, Abecassis PY, Vincent L, Nicolas JP, Lengauer C, Garcia-Echeverria C, Schio L.: Preparation and optimization of new 4-(2-(indolin-1-yl)-2-oxoethyl)-2-morpholinothiazole-5-carboxylic acid and amide derivatives as potent and selective PI3Kβ inhibitors. Bioorg Med Chem Lett, Volume 24 (6), 2014
Authors: Abecassis PY, Bertin L, Carry JC, Certal V, Charrier V, Filoche-Rommé B, Garcia-Echeverria C, Gruss-Leleu F, Guizani H, Halley F, Karlsson A, Lengauer C, Nicolas JP, Pilorge F, Richepin P, Schio L., Vincent L, Virone-Oddos A
Journal: Bioorg Med Chem Lett
Year: 2014
DOI: 10.1016/j.bmcl.2014.02.004
PubMed: 24560540
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