{"data":{"id":4005,"citation":"Certal V, Halley F, Virone-Oddos A, Filoche-Romm\u00e9 B, Carry JC, Gruss-Leleu F, Bertin L, Guizani H, Pilorge F, Richepin P, Karlsson A, Charrier V, Abecassis PY, Vincent L, Nicolas JP, Lengauer C, Garcia-Echeverria C, Schio L.: Preparation and optimization of new 4-(2-(indolin-1-yl)-2-oxoethyl)-2-morpholinothiazole-5-carboxylic acid and amide derivatives as potent and selective PI3K\u03b2 inhibitors. Bioorg Med Chem Lett, Volume 24 (6), 2014","title":"Preparation and optimization of new 4-(2-(indolin-1-yl)-2-oxoethyl)-2-morpholinothiazole-5-carboxylic acid and amide derivatives as potent and selective PI3K\u03b2 inhibitors.","doi":"10.1016\/j.bmcl.2014.02.004","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2014.02.004","pmid":"24560540","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/24560540\/","year":2014,"journal":"Bioorg Med Chem Lett","volume":"24","issue":"6","page":"1506-1510","authors":[{"first_name":"Abecassis PY","last_name":null,"full_name":null},{"first_name":"Bertin L","last_name":null,"full_name":null},{"first_name":"Carry JC","last_name":null,"full_name":null},{"first_name":"Certal V","last_name":null,"full_name":null},{"first_name":"Charrier V","last_name":null,"full_name":null},{"first_name":"Filoche-Romm\u00e9 B","last_name":null,"full_name":null},{"first_name":"Garcia-Echeverria C","last_name":null,"full_name":null},{"first_name":"Gruss-Leleu F","last_name":null,"full_name":null},{"first_name":"Guizani H","last_name":null,"full_name":null},{"first_name":"Halley F","last_name":null,"full_name":null},{"first_name":"Karlsson A","last_name":null,"full_name":null},{"first_name":"Lengauer C","last_name":null,"full_name":null},{"first_name":"Nicolas JP","last_name":null,"full_name":null},{"first_name":"Pilorge F","last_name":null,"full_name":null},{"first_name":"Richepin P","last_name":null,"full_name":null},{"first_name":"Schio L.","last_name":null,"full_name":null},{"first_name":"Vincent L","last_name":null,"full_name":null},{"first_name":"Virone-Oddos A","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/4005","landing_page":"https:\/\/molmedb.upol.cz\/publication\/4005","created_at":"2024-05-21T20:14:32.000000Z","updated_at":null}}