Discovery and Optimization of Orally Bioavailable Phthalazone and Cinnolone Carboxylic Acid Derivatives as S1P2 Antagonists against Fibrotic Diseases.

Publication

Citation
Mammoliti O, Jansen K, El Bkassiny S, Palisse A, Triballeau N, Bucher D, Allart B, Jaunet A, Tricarico G, De Wachter M, Menet C, Blanc J, Letfus V, Rupčić R, Šmehil M, Poljak T, Coornaert B, Sonck K, Duys I, Waeckel L, Lecru L, Marsais F, Jagerschmidt C, Auberval M, Pujuguet P, Oste L, Borgonovi M, Wakselman E, Christophe T, Houvenaghel N, Jans M, Heckmann B, Sanière L, Brys R.: Discovery and Optimization of Orally Bioavailable Phthalazone and Cinnolone Carboxylic Acid Derivatives as S1P2 Antagonists against Fibrotic Diseases. J Med Chem, Volume 64 (19), 2021
Authors
Allart B, Auberval M, Blanc J, Borgonovi M, Brys R., Bucher D, Christophe T, Coornaert B, De Wachter M, Duys I, El Bkassiny S, Heckmann B, Houvenaghel N, Jagerschmidt C, Jans M, Jansen K, Jaunet A, Lecru L, Letfus V, Mammoliti O, Marsais F, Menet C, Oste L, Palisse A, Poljak T, Pujuguet P, Rupčić R, Saniere L, Šmehil M, Sonck K, Triballeau N, Tricarico G, Waeckel L, Wakselman E
Journal
J Med Chem
Year
2021
PubMed
34581584
Machine-readable
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Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

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  • MolMeDB interoperability with UniProt and SwissLipids – MEYS Czech-Swiss project ELIXIR-IMPACT 8K0208 (2026–2028)
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