{"data":{"id":3660,"citation":"Mammoliti O, Jansen K, El Bkassiny S, Palisse A, Triballeau N, Bucher D, Allart B, Jaunet A, Tricarico G, De Wachter M, Menet C, Blanc J, Letfus V, Rup\u010di\u0107 R, \u0160mehil M, Poljak T, Coornaert B, Sonck K, Duys I, Waeckel L, Lecru L, Marsais F, Jagerschmidt C, Auberval M, Pujuguet P, Oste L, Borgonovi M, Wakselman E, Christophe T, Houvenaghel N, Jans M, Heckmann B, Sani\u00e8re L, Brys R.: Discovery and Optimization of Orally Bioavailable Phthalazone and Cinnolone Carboxylic Acid Derivatives as S1P2 Antagonists against Fibrotic Diseases. J Med Chem, Volume 64 (19), 2021","title":"Discovery and Optimization of Orally Bioavailable Phthalazone and Cinnolone Carboxylic Acid Derivatives as S1P2 Antagonists against Fibrotic Diseases.","doi":"10.1021\/acs.jmedchem.1c01066","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.1c01066","pmid":"34581584","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/34581584\/","year":2021,"journal":"J Med Chem","volume":"64","issue":"19","page":"14557-14586","authors":[{"first_name":"Allart B","last_name":null,"full_name":null},{"first_name":"Auberval M","last_name":null,"full_name":null},{"first_name":"Blanc J","last_name":null,"full_name":null},{"first_name":"Borgonovi M","last_name":null,"full_name":null},{"first_name":"Brys R.","last_name":null,"full_name":null},{"first_name":"Bucher D","last_name":null,"full_name":null},{"first_name":"Christophe T","last_name":null,"full_name":null},{"first_name":"Coornaert B","last_name":null,"full_name":null},{"first_name":"De Wachter M","last_name":null,"full_name":null},{"first_name":"Duys I","last_name":null,"full_name":null},{"first_name":"El Bkassiny S","last_name":null,"full_name":null},{"first_name":"Heckmann B","last_name":null,"full_name":null},{"first_name":"Houvenaghel N","last_name":null,"full_name":null},{"first_name":"Jagerschmidt C","last_name":null,"full_name":null},{"first_name":"Jans M","last_name":null,"full_name":null},{"first_name":"Jansen K","last_name":null,"full_name":null},{"first_name":"Jaunet A","last_name":null,"full_name":null},{"first_name":"Lecru L","last_name":null,"full_name":null},{"first_name":"Letfus V","last_name":null,"full_name":null},{"first_name":"Mammoliti O","last_name":null,"full_name":null},{"first_name":"Marsais F","last_name":null,"full_name":null},{"first_name":"Menet C","last_name":null,"full_name":null},{"first_name":"Oste L","last_name":null,"full_name":null},{"first_name":"Palisse A","last_name":null,"full_name":null},{"first_name":"Poljak T","last_name":null,"full_name":null},{"first_name":"Pujuguet P","last_name":null,"full_name":null},{"first_name":"Rup\u010di\u0107 R","last_name":null,"full_name":null},{"first_name":"Saniere L","last_name":null,"full_name":null},{"first_name":"\u0160mehil M","last_name":null,"full_name":null},{"first_name":"Sonck K","last_name":null,"full_name":null},{"first_name":"Triballeau N","last_name":null,"full_name":null},{"first_name":"Tricarico G","last_name":null,"full_name":null},{"first_name":"Waeckel L","last_name":null,"full_name":null},{"first_name":"Wakselman E","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3660","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3660","created_at":"2024-05-21T20:12:51.000000Z","updated_at":null}}