Citation

Shi Q, Xiao Z, Yang MG, Marcoux D, Cherney RJ, Yip S, Li P, Wu DR, Weigelt CA, Sack J, Khan J, Ruzanov M, Wang J, Yarde M, Ellen Cvijic M, Li S, Shuster DJ, Xie J, Sherry T, Obermeier M, Fura A, Stefanski K, Cornelius G, Chacko S, Shu YZ, Khandelwal P, Hynes J, Tino JA, Salter-Cid L, Denton R, Zhao Q, Dhar TGM.: Tricyclic sulfones as potent, selective and efficacious RORγt inverse agonists - Exploring C6 and C8 SAR using late-stage functionalization. Bioorg Med Chem Lett, Volume 30 (23), 2020

Authors

Chacko S, Cherney RJ, Cornelius G, Denton R, Dhar TGM., Ellen Cvijic M, Fura A, Hynes J, Khan J, Khandelwal P, Li P, Li S, Marcoux D, Obermeier M, Ruzanov M, Sack J, Salter-Cid L, Sherry T, Shi Q, Shu YZ, Shuster DJ, Stefanski K, Tino JA, Wang J, Weigelt CA, Wu DR, Xiao Z, Xie J, Yang MG, Yarde M, Yip S, Zhao Q

Journal

Bioorg Med Chem Lett

Year

2020

DOI

10.1016/j.bmcl.2020.127521

PubMed

32882417

Machine-readable

REST APIRDF