{"data":{"id":3651,"citation":"Shi Q, Xiao Z, Yang MG, Marcoux D, Cherney RJ, Yip S, Li P, Wu DR, Weigelt CA, Sack J, Khan J, Ruzanov M, Wang J, Yarde M, Ellen Cvijic M, Li S, Shuster DJ, Xie J, Sherry T, Obermeier M, Fura A, Stefanski K, Cornelius G, Chacko S, Shu YZ, Khandelwal P, Hynes J, Tino JA, Salter-Cid L, Denton R, Zhao Q, Dhar TGM.: Tricyclic sulfones as potent, selective and efficacious ROR\u03b3t inverse agonists - Exploring C6 and C8 SAR using late-stage functionalization. Bioorg Med Chem Lett, Volume 30 (23), 2020","title":"Tricyclic sulfones as potent, selective and efficacious ROR\u03b3t inverse agonists - Exploring C6 and C8 SAR using late-stage functionalization.","doi":"10.1016\/j.bmcl.2020.127521","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2020.127521","pmid":"32882417","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/32882417\/","year":2020,"journal":"Bioorg Med Chem Lett","volume":"30","issue":"23","page":"127521","authors":[{"first_name":"Chacko S","last_name":null,"full_name":null},{"first_name":"Cherney RJ","last_name":null,"full_name":null},{"first_name":"Cornelius G","last_name":null,"full_name":null},{"first_name":"Denton R","last_name":null,"full_name":null},{"first_name":"Dhar TGM.","last_name":null,"full_name":null},{"first_name":"Ellen Cvijic M","last_name":null,"full_name":null},{"first_name":"Fura A","last_name":null,"full_name":null},{"first_name":"Hynes J","last_name":null,"full_name":null},{"first_name":"Khan J","last_name":null,"full_name":null},{"first_name":"Khandelwal P","last_name":null,"full_name":null},{"first_name":"Li P","last_name":null,"full_name":null},{"first_name":"Li S","last_name":null,"full_name":null},{"first_name":"Marcoux D","last_name":null,"full_name":null},{"first_name":"Obermeier M","last_name":null,"full_name":null},{"first_name":"Ruzanov M","last_name":null,"full_name":null},{"first_name":"Sack J","last_name":null,"full_name":null},{"first_name":"Salter-Cid L","last_name":null,"full_name":null},{"first_name":"Sherry T","last_name":null,"full_name":null},{"first_name":"Shi Q","last_name":null,"full_name":null},{"first_name":"Shu YZ","last_name":null,"full_name":null},{"first_name":"Shuster DJ","last_name":null,"full_name":null},{"first_name":"Stefanski K","last_name":null,"full_name":null},{"first_name":"Tino JA","last_name":null,"full_name":null},{"first_name":"Wang J","last_name":null,"full_name":null},{"first_name":"Weigelt CA","last_name":null,"full_name":null},{"first_name":"Wu DR","last_name":null,"full_name":null},{"first_name":"Xiao Z","last_name":null,"full_name":null},{"first_name":"Xie J","last_name":null,"full_name":null},{"first_name":"Yang MG","last_name":null,"full_name":null},{"first_name":"Yarde M","last_name":null,"full_name":null},{"first_name":"Yip S","last_name":null,"full_name":null},{"first_name":"Zhao Q","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3651","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3651","created_at":"2024-05-21T20:12:50.000000Z","updated_at":null}}