Citation

Moslin R, Zhang Y, Wrobleski ST, Lin S, Mertzman M, Spergel S, Tokarski JS, Strnad J, Gillooly K, McIntyre KW, Zupa-Fernandez A, Cheng L, Sun H, Chaudhry C, Huang C, D'Arienzo C, Heimrich E, Yang X, Muckelbauer JK, Chang C, Tredup J, Mulligan D, Xie D, Aranibar N, Chiney M, Burke JR, Lombardo L, Carter PH, Weinstein DS.: Identification of <i>N</i>-Methyl Nicotinamide and <i>N</i>-Methyl Pyridazine-3-Carboxamide Pseudokinase Domain Ligands as Highly Selective Allosteric Inhibitors of Tyrosine Kinase 2 (TYK2). J Med Chem, Volume 62 (20), 2019

Authors

Aranibar N, Burke JR, Carter PH, Chang C, Chaudhry C, Cheng L, Chiney M, D'Arienzo C, Gillooly K, Heimrich E, Huang C, Lin S, Lombardo L, McIntyre KW, Mertzman M, Moslin R, Muckelbauer JK, Mulligan D, Spergel S, Strnad J, Sun H, Tokarski JS, Tredup J, Weinstein DS., Wrobleski ST, Xie D, Yang X, Zhang Y, Zupa-Fernandez A

Journal

J Med Chem

Year

2019

DOI

10.1021/acs.jmedchem.9b00443

PubMed

31314518

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