{"data":{"id":3382,"citation":"Moslin R, Zhang Y, Wrobleski ST, Lin S, Mertzman M, Spergel S, Tokarski JS, Strnad J, Gillooly K, McIntyre KW, Zupa-Fernandez A, Cheng L, Sun H, Chaudhry C, Huang C, D'Arienzo C, Heimrich E, Yang X, Muckelbauer JK, Chang C, Tredup J, Mulligan D, Xie D, Aranibar N, Chiney M, Burke JR, Lombardo L, Carter PH, Weinstein DS.: Identification of <i>N<\/i>-Methyl Nicotinamide and <i>N<\/i>-Methyl Pyridazine-3-Carboxamide Pseudokinase Domain Ligands as Highly Selective Allosteric Inhibitors of Tyrosine Kinase 2 (TYK2). J Med Chem, Volume 62 (20), 2019","title":"Identification of <i>N<\/i>-Methyl Nicotinamide and <i>N<\/i>-Methyl Pyridazine-3-Carboxamide Pseudokinase Domain Ligands as Highly Selective Allosteric Inhibitors of Tyrosine Kinase 2 (TYK2).","doi":"10.1021\/acs.jmedchem.9b00443","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.9b00443","pmid":"31314518","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/31314518\/","year":2019,"journal":"J Med Chem","volume":"62","issue":"20","page":"8953-8972","authors":[{"first_name":"Aranibar N","last_name":null,"full_name":null},{"first_name":"Burke JR","last_name":null,"full_name":null},{"first_name":"Carter PH","last_name":null,"full_name":null},{"first_name":"Chang C","last_name":null,"full_name":null},{"first_name":"Chaudhry C","last_name":null,"full_name":null},{"first_name":"Cheng L","last_name":null,"full_name":null},{"first_name":"Chiney M","last_name":null,"full_name":null},{"first_name":"D'Arienzo C","last_name":null,"full_name":null},{"first_name":"Gillooly K","last_name":null,"full_name":null},{"first_name":"Heimrich E","last_name":null,"full_name":null},{"first_name":"Huang C","last_name":null,"full_name":null},{"first_name":"Lin S","last_name":null,"full_name":null},{"first_name":"Lombardo L","last_name":null,"full_name":null},{"first_name":"McIntyre KW","last_name":null,"full_name":null},{"first_name":"Mertzman M","last_name":null,"full_name":null},{"first_name":"Moslin R","last_name":null,"full_name":null},{"first_name":"Muckelbauer JK","last_name":null,"full_name":null},{"first_name":"Mulligan D","last_name":null,"full_name":null},{"first_name":"Spergel S","last_name":null,"full_name":null},{"first_name":"Strnad J","last_name":null,"full_name":null},{"first_name":"Sun H","last_name":null,"full_name":null},{"first_name":"Tokarski JS","last_name":null,"full_name":null},{"first_name":"Tredup J","last_name":null,"full_name":null},{"first_name":"Weinstein DS.","last_name":null,"full_name":null},{"first_name":"Wrobleski ST","last_name":null,"full_name":null},{"first_name":"Xie D","last_name":null,"full_name":null},{"first_name":"Yang X","last_name":null,"full_name":null},{"first_name":"Zhang Y","last_name":null,"full_name":null},{"first_name":"Zupa-Fernandez A","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/3382","landing_page":"https:\/\/molmedb.upol.cz\/publication\/3382","created_at":"2024-05-21T20:11:53.000000Z","updated_at":null}}