Citation

Wang L, Pratt JK, Soltwedel T, Sheppard GS, Fidanze SD, Liu D, Hasvold LA, Mantei RA, Holms JH, McClellan WJ, Wendt MD, Wada C, Frey R, Hansen TM, Hubbard R, Park CH, Li L, Magoc TJ, Albert DH, Lin X, Warder SE, Kovar P, Huang X, Wilcox D, Wang R, Rajaraman G, Petros AM, Hutchins CW, Panchal SC, Sun C, Elmore SW, Shen Y, Kati WM, McDaniel KF.: Fragment-Based, Structure-Enabled Discovery of Novel Pyridones and Pyridone Macrocycles as Potent Bromodomain and Extra-Terminal Domain (BET) Family Bromodomain Inhibitors. J Med Chem, Volume 60 (9), 2017

Authors

Albert DH, Elmore SW, Fidanze SD, Frey R, Hansen TM, Hasvold LA, Holms JH, Huang X, Hubbard R, Hutchins CW, Kati WM, Kovar P, Li L, Lin X, Liu D, Magoc TJ, Mantei RA, McClellan WJ, McDaniel KF., Panchal SC, Park CH, Petros AM, Pratt JK, Rajaraman G, Shen Y, Sheppard GS, Soltwedel T, Sun C, Wada C, Wang L, Wang R, Warder SE, Wendt MD, Wilcox D

Journal

J Med Chem

Year

2017

DOI

10.1021/acs.jmedchem.7b00017

PubMed

28368119

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