{"data":{"id":2717,"citation":"Wang L, Pratt JK, Soltwedel T, Sheppard GS, Fidanze SD, Liu D, Hasvold LA, Mantei RA, Holms JH, McClellan WJ, Wendt MD, Wada C, Frey R, Hansen TM, Hubbard R, Park CH, Li L, Magoc TJ, Albert DH, Lin X, Warder SE, Kovar P, Huang X, Wilcox D, Wang R, Rajaraman G, Petros AM, Hutchins CW, Panchal SC, Sun C, Elmore SW, Shen Y, Kati WM, McDaniel KF.: Fragment-Based, Structure-Enabled Discovery of Novel Pyridones and Pyridone Macrocycles as Potent Bromodomain and Extra-Terminal Domain (BET) Family Bromodomain Inhibitors. J Med Chem, Volume 60 (9), 2017","title":"Fragment-Based, Structure-Enabled Discovery of Novel Pyridones and Pyridone Macrocycles as Potent Bromodomain and Extra-Terminal Domain (BET) Family Bromodomain Inhibitors.","doi":"10.1021\/acs.jmedchem.7b00017","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.7b00017","pmid":"28368119","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/28368119\/","year":2017,"journal":"J Med Chem","volume":"60","issue":"9","page":"3828-3850","authors":[{"first_name":"Albert DH","last_name":null,"full_name":null},{"first_name":"Elmore SW","last_name":null,"full_name":null},{"first_name":"Fidanze SD","last_name":null,"full_name":null},{"first_name":"Frey R","last_name":null,"full_name":null},{"first_name":"Hansen TM","last_name":null,"full_name":null},{"first_name":"Hasvold LA","last_name":null,"full_name":null},{"first_name":"Holms JH","last_name":null,"full_name":null},{"first_name":"Huang X","last_name":null,"full_name":null},{"first_name":"Hubbard R","last_name":null,"full_name":null},{"first_name":"Hutchins CW","last_name":null,"full_name":null},{"first_name":"Kati WM","last_name":null,"full_name":null},{"first_name":"Kovar P","last_name":null,"full_name":null},{"first_name":"Li L","last_name":null,"full_name":null},{"first_name":"Lin X","last_name":null,"full_name":null},{"first_name":"Liu D","last_name":null,"full_name":null},{"first_name":"Magoc TJ","last_name":null,"full_name":null},{"first_name":"Mantei RA","last_name":null,"full_name":null},{"first_name":"McClellan WJ","last_name":null,"full_name":null},{"first_name":"McDaniel KF.","last_name":null,"full_name":null},{"first_name":"Panchal SC","last_name":null,"full_name":null},{"first_name":"Park CH","last_name":null,"full_name":null},{"first_name":"Petros AM","last_name":null,"full_name":null},{"first_name":"Pratt JK","last_name":null,"full_name":null},{"first_name":"Rajaraman G","last_name":null,"full_name":null},{"first_name":"Shen Y","last_name":null,"full_name":null},{"first_name":"Sheppard GS","last_name":null,"full_name":null},{"first_name":"Soltwedel T","last_name":null,"full_name":null},{"first_name":"Sun C","last_name":null,"full_name":null},{"first_name":"Wada C","last_name":null,"full_name":null},{"first_name":"Wang L","last_name":null,"full_name":null},{"first_name":"Wang R","last_name":null,"full_name":null},{"first_name":"Warder SE","last_name":null,"full_name":null},{"first_name":"Wendt MD","last_name":null,"full_name":null},{"first_name":"Wilcox D","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2717","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2717","created_at":"2023-06-23T15:09:27.000000Z","updated_at":null}}