- Citation
- Sakauchi N, Kohara Y, Sato A, Suzaki T, Imai Y, Okabe Y, Imai S, Saikawa R, Nagabukuro H, Kuno H, Fujita H, Kamo I, Yoshida M.: Discovery of 5-Chloro-1-(5-chloro-2-(methylsulfonyl)benzyl)-2-imino-1,2-dihydropyridine-3-carboxamide (TAK-259) as a Novel, Selective, and Orally Active α1D Adrenoceptor Antagonist with Antiurinary Frequency Effects: Reducing Human Ether-a-go-go-Related Gene (hERG) Liabilities. J Med Chem, Volume 59 (7), 2016
- Authors
- Fujita H, Imai S, Imai Y, Kamo I, Kohara Y, Kuno H, Nagabukuro H, Okabe Y, Saikawa R, Sakauchi N, Sato A, Suzaki T, Yoshida M.
- Journal
- J Med Chem
- Year
- 2016
- Machine-readable
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