Design and synthesis of hydroxyethylamine (HEA) BACE-1 inhibitors: structure-activity relationship of the aryl region.

Publication

Citation
Probst GD, Bowers S, Sealy JM, Stupi B, Dressen D, Jagodzinska BM, Aquino J, Gailunas A, Truong AP, Tso L, Xu YZ, Hom RK, John V, Tung JS, Pleiss MA, Tucker JA, Konradi AW, Sham HL, Jagodzinski J, Toth G, Brecht E, Yao N, Pan H, Lin M, Artis DR, Ruslim L, Bova MP, Sinha S, Yednock TA, Gauby S, Zmolek W, Quinn KP, Sauer JM.: Design and synthesis of hydroxyethylamine (HEA) BACE-1 inhibitors: structure-activity relationship of the aryl region. Bioorg Med Chem Lett, Volume 20 (20), 2010
Authors
Aquino J, Artis DR, Bova MP, Bowers S, Brecht E, Dressen D, Gailunas A, Gauby S, Hom RK, Jagodzinska BM, Jagodzinski J, John V, Konradi AW, Lin M, Pan H, Pleiss MA, Probst GD, Quinn KP, Ruslim L, Sauer JM., Sealy JM, Sham HL, Sinha S, Stupi B, Toth G, Truong AP, Tso L, Tucker JA, Tung JS, Xu YZ, Yao N, Yednock TA, Zmolek W
Journal
Bioorg Med Chem Lett
Year
2010
PubMed
20822903
Machine-readable
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Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

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