{"data":{"id":2289,"citation":"Probst GD, Bowers S, Sealy JM, Stupi B, Dressen D, Jagodzinska BM, Aquino J, Gailunas A, Truong AP, Tso L, Xu YZ, Hom RK, John V, Tung JS, Pleiss MA, Tucker JA, Konradi AW, Sham HL, Jagodzinski J, Toth G, Brecht E, Yao N, Pan H, Lin M, Artis DR, Ruslim L, Bova MP, Sinha S, Yednock TA, Gauby S, Zmolek W, Quinn KP, Sauer JM.: Design and synthesis of hydroxyethylamine (HEA) BACE-1 inhibitors: structure-activity relationship of the aryl region. Bioorg Med Chem Lett, Volume 20 (20), 2010","title":"Design and synthesis of hydroxyethylamine (HEA) BACE-1 inhibitors: structure-activity relationship of the aryl region.","doi":"10.1016\/j.bmcl.2010.08.070","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2010.08.070","pmid":"20822903","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/20822903\/","year":2010,"journal":"Bioorg Med Chem Lett","volume":"20","issue":"20","page":"6034-6039","authors":[{"first_name":"Aquino J","last_name":null,"full_name":null},{"first_name":"Artis DR","last_name":null,"full_name":null},{"first_name":"Bova MP","last_name":null,"full_name":null},{"first_name":"Bowers S","last_name":null,"full_name":null},{"first_name":"Brecht E","last_name":null,"full_name":null},{"first_name":"Dressen D","last_name":null,"full_name":null},{"first_name":"Gailunas A","last_name":null,"full_name":null},{"first_name":"Gauby S","last_name":null,"full_name":null},{"first_name":"Hom RK","last_name":null,"full_name":null},{"first_name":"Jagodzinska BM","last_name":null,"full_name":null},{"first_name":"Jagodzinski J","last_name":null,"full_name":null},{"first_name":"John V","last_name":null,"full_name":null},{"first_name":"Konradi AW","last_name":null,"full_name":null},{"first_name":"Lin M","last_name":null,"full_name":null},{"first_name":"Pan H","last_name":null,"full_name":null},{"first_name":"Pleiss MA","last_name":null,"full_name":null},{"first_name":"Probst GD","last_name":null,"full_name":null},{"first_name":"Quinn KP","last_name":null,"full_name":null},{"first_name":"Ruslim L","last_name":null,"full_name":null},{"first_name":"Sauer JM.","last_name":null,"full_name":null},{"first_name":"Sealy JM","last_name":null,"full_name":null},{"first_name":"Sham HL","last_name":null,"full_name":null},{"first_name":"Sinha S","last_name":null,"full_name":null},{"first_name":"Stupi B","last_name":null,"full_name":null},{"first_name":"Toth G","last_name":null,"full_name":null},{"first_name":"Truong AP","last_name":null,"full_name":null},{"first_name":"Tso L","last_name":null,"full_name":null},{"first_name":"Tucker JA","last_name":null,"full_name":null},{"first_name":"Tung JS","last_name":null,"full_name":null},{"first_name":"Xu YZ","last_name":null,"full_name":null},{"first_name":"Yao N","last_name":null,"full_name":null},{"first_name":"Yednock TA","last_name":null,"full_name":null},{"first_name":"Zmolek W","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/2289","landing_page":"https:\/\/molmedb.upol.cz\/publication\/2289","created_at":"2023-06-23T10:46:17.000000Z","updated_at":null}}