- Citation
- Koltun DO, Parkhill EQ, Elzein E, Kobayashi T, Jiang RH, Li X, Perry TD, Avila B, Wang WQ, Hirakawa R, Smith-Maxwell C, Wu L, Dhalla AK, Rajamani S, Mollova N, Stafford B, Tang J, Belardinelli L, Zablocki JA.: Discovery of triazolopyridinone GS-462808, a late sodium current inhibitor (Late INai) of the cardiac Nav1.5 channel with improved efficacy and potency relative to ranolazine. Bioorg Med Chem Lett, Volume 26 (13), 2016
- Authors
- Avila B, Belardinelli L, Dhalla AK, Elzein E, Hirakawa R, Jiang RH, Kobayashi T, Koltun DO, Li X, Mollova N, Parkhill EQ, Perry TD, Rajamani S, Smith-Maxwell C, Stafford B, Tang J, Wang WQ, Wu L, Zablocki JA.
- Journal
- Bioorg Med Chem Lett
- Year
- 2016
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