{"data":{"id":1489,"citation":"Koltun DO, Parkhill EQ, Elzein E, Kobayashi T, Jiang RH, Li X, Perry TD, Avila B, Wang WQ, Hirakawa R, Smith-Maxwell C, Wu L, Dhalla AK, Rajamani S, Mollova N, Stafford B, Tang J, Belardinelli L, Zablocki JA.: Discovery of triazolopyridinone GS-462808, a late sodium current inhibitor (Late INai) of the cardiac Nav1.5 channel with improved efficacy and potency relative to ranolazine. Bioorg Med Chem Lett, Volume 26 (13), 2016","title":"Discovery of triazolopyridinone GS-462808, a late sodium current inhibitor (Late INai) of the cardiac Nav1.5 channel with improved efficacy and potency relative to ranolazine.","doi":"10.1016\/j.bmcl.2016.03.096","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2016.03.096","pmid":"27038498","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/27038498\/","year":2016,"journal":"Bioorg Med Chem Lett","volume":"26","issue":"13","page":"3207-3211","authors":[{"first_name":"Avila B","last_name":null,"full_name":null},{"first_name":"Belardinelli L","last_name":null,"full_name":null},{"first_name":"Dhalla AK","last_name":null,"full_name":null},{"first_name":"Elzein E","last_name":null,"full_name":null},{"first_name":"Hirakawa R","last_name":null,"full_name":null},{"first_name":"Jiang RH","last_name":null,"full_name":null},{"first_name":"Kobayashi T","last_name":null,"full_name":null},{"first_name":"Koltun DO","last_name":null,"full_name":null},{"first_name":"Li X","last_name":null,"full_name":null},{"first_name":"Mollova N","last_name":null,"full_name":null},{"first_name":"Parkhill EQ","last_name":null,"full_name":null},{"first_name":"Perry TD","last_name":null,"full_name":null},{"first_name":"Rajamani S","last_name":null,"full_name":null},{"first_name":"Smith-Maxwell C","last_name":null,"full_name":null},{"first_name":"Stafford B","last_name":null,"full_name":null},{"first_name":"Tang J","last_name":null,"full_name":null},{"first_name":"Wang WQ","last_name":null,"full_name":null},{"first_name":"Wu L","last_name":null,"full_name":null},{"first_name":"Zablocki JA.","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/1489","landing_page":"https:\/\/molmedb.upol.cz\/publication\/1489","created_at":"2021-01-20T12:16:54.000000Z","updated_at":null}}