Discovery and hit-to-lead optimization of pyrrolopyrimidines as potent, state-dependent Na(v)1.7 antagonists.

Publication

Citation
Chakka N, Bregman H, Du B, Nguyen HN, Buchanan JL, Feric E, Ligutti J, Liu D, McDermott JS, Zou A, McDonough SI, Dimauro EF.: Discovery and hit-to-lead optimization of pyrrolopyrimidines as potent, state-dependent Na(v)1.7 antagonists. Bioorg Med Chem Lett, Volume 22 (5), 2012
Authors
Bregman H, Buchanan JL, Chakka N, Dimauro EF., Du B, Feric E, Ligutti J, Liu D, McDermott JS, McDonough SI, Nguyen HN, Zou A
Journal
Bioorg Med Chem Lett
Year
2012
PubMed
22318156
Machine-readable
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Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

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