- Citation
- Koltun DO, Parkhill EQ, Elzein E, Kobayashi T, Notte GT, Kalla R, Jiang RH, Li X, Perry TD, Avila B, Wang WQ, Smith-Maxwell C, Dhalla AK, Rajamani S, Stafford B, Tang J, Mollova N, Belardinelli L, Zablocki JA.: Discovery of triazolopyridine GS-458967, a late sodium current inhibitor (Late INai) of the cardiac NaV 1.5 channel with improved efficacy and potency relative to ranolazine. Bioorg Med Chem Lett, Volume 26 (13), 2016
- Authors
- Avila B, Belardinelli L, Dhalla AK, Elzein E, Jiang RH, Kalla R, Kobayashi T, Koltun DO, Li X, Mollova N, Notte GT, Parkhill EQ, Perry TD, Rajamani S, Smith-Maxwell C, Stafford B, Tang J, Wang WQ, Zablocki JA.
- Journal
- Bioorg Med Chem Lett
- Year
- 2016
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