- Citation
- Focken T, Chowdhury S, Zenova A, Grimwood ME, Chabot C, Sheng T, Hemeon I, Decker SM, Wilson M, Bichler P, Jia Q, Sun S, Young C, Lin S, Goodchild SJ, Shuart NG, Chang E, Xie Z, Li B, Khakh K, Bankar G, Waldbrook M, Kwan R, Nelkenbrecher K, Karimi Tari P, Chahal N, Sojo L, Robinette CL, White AD, Chen CA, Zhang Y, Pang J, Chang JH, Hackos DH, Johnson JP, Cohen CJ, Ortwine DF, Sutherlin DP, Dehnhardt CM, Safina BS.: Design of Conformationally Constrained Acyl Sulfonamide Isosteres: Identification of N-([1,2,4]Triazolo[4,3- a]pyridin-3-yl)methane-sulfonamides as Potent and Selective hNaV1.7 Inhibitors for the Treatment of Pain. J Med Chem, Volume 61 (11), 2018
- Authors
- Bankar G, Bichler P, Chabot C, Chahal N, Chang E, Chang JH, Chen CA, Chowdhury S, Decker SM, Focken T, Goodchild SJ, Grimwood ME, Hackos DH, Hemeon I, Jia Q, Karimi Tari P, Khakh K, Kwan R, Li B, Lin S, Nelkenbrecher K, Pang J, Robinette CL, Sheng T, Shuart NG, Sojo L, Sun S, Waldbrook M, White AD, Wilson M, Xie Z, Young C, Zenova A, Zhang Y, Cohen CJ, Dehnhardt CM, Johnson JP, Ortwine DF, Safina BS., Sutherlin DP
- Journal
- J Med Chem
- Year
- 2018
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