Citation

Luo G, Chen L, Kostich WA, Hamman B, Allen J, Easton A, Bourin C, Gulianello M, Lippy J, Nara S, Pattipati SN, Dandapani K, Dokania M, Vattikundala P, Sharma V, Elavazhagan S, Verma MK, Lal Das M, Wagh S, Balakrishnan A, Johnson BM, Santone KS, Thalody G, Denton R, Saminathan H, Holenarsipur VK, Kumar A, Rao A, Putlur SP, Sarvasiddhi SK, Shankar G, Louis JV, Ramarao M, Conway CM, Li YW, Pieschl R, Tian Y, Hong Y, Bristow L, Albright CF, Bronson JJ, Macor JE, Dzierba CD.: Discovery and Optimization of Biaryl Alkyl Ethers as a Novel Class of Highly Selective, CNS-Penetrable, and Orally Active Adaptor Protein-2-Associated Kinase 1 (AAK1) Inhibitors for the Potential Treatment of Neuropathic Pain. J Med Chem, Volume 65 (6), 2022

Authors

Albright CF, Allen J, Balakrishnan A, Bourin C, Bristow L, Bronson JJ, Chen L, Conway CM, Dandapani K, Denton R, Dokania M, Dzierba CD., Easton A, Elavazhagan S, Gulianello M, Hamman B, Holenarsipur VK, Hong Y, Johnson BM, Kostich WA, Kumar A, Lal Das M, Li YW, Lippy J, Louis JV, Luo G, Macor JE, Nara S, Pattipati SN, Pieschl R, Putlur SP, Ramarao M, Rao A, Saminathan H, Santone KS, Sarvasiddhi SK, Shankar G, Sharma V, Thalody G, Tian Y, Vattikundala P, Verma MK, Wagh S

Journal

J Med Chem

Year

2022

DOI

10.1021/acs.jmedchem.1c02132

PubMed

35261239

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