- Citation
- De Lucca GV, Shi Q, Liu Q, Batt DG, Beaudoin Bertrand M, Rampulla R, Mathur A, Discenza L, D'Arienzo C, Dai J, Obermeier M, Vickery R, Zhang Y, Yang Z, Marathe P, Tebben AJ, Muckelbauer JK, Chang CJ, Zhang H, Gillooly K, Taylor T, Pattoli MA, Skala S, Kukral DW, McIntyre KW, Salter-Cid L, Fura A, Burke JR, Barrish JC, Carter PH, Tino JA.: Small Molecule Reversible Inhibitors of Bruton's Tyrosine Kinase (BTK): Structure-Activity Relationships Leading to the Identification of 7-(2-Hydroxypropan-2-yl)-4-[2-methyl-3-(4-oxo-3,4-dihydroquinazolin-3-yl)phenyl]-9H-carbazole-1-carboxamide (BMS-935177). J Med Chem, Volume 59 (17), 2016
- Authors
- Barrish JC, Batt DG, Beaudoin Bertrand M, Burke JR, Carter PH, Chang CJ, D'Arienzo C, Dai J, De Lucca GV, Discenza L, Fura A, Gillooly K, Kukral DW, Liu Q, Marathe P, Mathur A, McIntyre KW, Muckelbauer JK, Obermeier M, Pattoli MA, Rampulla R, Salter-Cid L, Shi Q, Skala S, Taylor T, Tebben AJ, Tino JA., Vickery R, Yang Z, Zhang H, Zhang Y
- Journal
- J Med Chem
- Year
- 2016
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