Discovery and Optimization of a Series of Benzofuran Selective ERAP1 Inhibitors: Biochemical and <i>In Silico</i> Studies.

Publication

Citation
Deddouche-Grass S, Andouche C, Bärenz F, Halter C, Hohwald A, Lebrun L, Membré N, Morales R, Muzet N, Poirot M, Reynaud M, Roujean V, Weber F, Zimmermann A, Heng R, Basse N.: Discovery and Optimization of a Series of Benzofuran Selective ERAP1 Inhibitors: Biochemical and <i>In Silico</i> Studies. ACS Med Chem Lett, Volume 12 (7), 2021
Authors
Andouche C, Bärenz F, Basse N., Deddouche-Grass S, Halter C, Heng R, Hohwald A, LeBrun L, Membré N, Morales R, Muzet N, Poirot M, Reynaud M, Roujean V, Weber F, Zimmermann A
Journal
ACS Med Chem Lett
Year
2021
PubMed
34267884
Machine-readable
REST APIRDF
Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

Follow us

FacebookGithub

Financial Support

  • MolMeDB interoperability with UniProt and SwissLipids – MEYS Czech-Swiss project ELIXIR-IMPACT 8K0208 (2026–2028)
ELIXIRGAČRUP Olomouc