Novel N-linked aminopiperidine-based gyrase inhibitors with improved hERG and in vivo efficacy against Mycobacterium tuberculosis.

Publication

Citation
Hameed P S, Patil V, Solapure S, Sharma U, Madhavapeddi P, Raichurkar A, Chinnapattu M, Manjrekar P, Shanbhag G, Puttur J, Shinde V, Menasinakai S, Rudrapatana S, Achar V, Awasthy D, Nandishaiah R, Humnabadkar V, Ghosh A, Narayan C, Ramya VK, Kaur P, Sharma S, Werngren J, Hoffner S, Panduga V, Kumar CN, Reddy J, Kumar K N M, Ganguly S, Bharath S, Bheemarao U, Mukherjee K, Arora U, Gaonkar S, Coulson M, Waterson D, Sambandamurthy VK, de Sousa SM.: Novel N-linked aminopiperidine-based gyrase inhibitors with improved hERG and in vivo efficacy against Mycobacterium tuberculosis. J Med Chem, Volume 57 (11), 2014
Authors
Achar V, Arora U, Awasthy D, Bharath S, Bheemarao U, Chinnapattu M, Coulson M, de Sousa SM., Ganguly S, Gaonkar S, Ghosh A, Hameed P S, Hoffner S, Humnabadkar V, Kaur P, Kumar CN, Kumar K N M, Madhavapeddi P, Manjrekar P, Menasinakai S, Mukherjee K, Nandishaiah R, Narayan C, Panduga V, Patil V, Puttur J, Raichurkar A, Ramya VK, Reddy J, Rudrapatana S, Sambandamurthy VK, Shanbhag G, Sharma S, Sharma U, Shinde V, Solapure S, Waterson D, Werngren J
Journal
J Med Chem
Year
2014
PubMed
24809953
Machine-readable
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Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

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