Discovery of Potent, Highly Selective, and <i>In Vivo</i> Efficacious, Allosteric MALT1 Inhibitors by Iterative Scaffold Morphing.

Publication

Citation
Pissot Soldermann C, Simic O, Renatus M, Erbel P, Melkko S, Wartmann M, Bigaud M, Weiss A, McSheehy P, Endres R, Santos P, Blank J, Schuffenhauer A, Bold G, Buschmann N, Zoller T, Altmann E, Manley PW, Dix I, Buchdunger E, Scesa J, Quancard J, Schlapbach A, Bornancin F, Radimerski T, Régnier CH.: Discovery of Potent, Highly Selective, and <i>In Vivo</i> Efficacious, Allosteric MALT1 Inhibitors by Iterative Scaffold Morphing. J Med Chem, Volume 63 (23), 2020
Authors
Altmann E, Bigaud M, Blank J, Bold G, Bornancin F, Buchdunger E, Buschmann N, Dix I, Endres R, Erbel P, Manley PW, Mcsheehy P, Melkko S, Pissot Soldermann C, Quancard J, Radimerski T, Régnier CH., Renatus M, Santos P, Scesa J, Schlapbach A, Schuffenhauer A, Simic O, Wartmann M, Weiss A, Zoller T
Journal
J Med Chem
Year
2020
PubMed
33252239
Machine-readable
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Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

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  • MolMeDB interoperability with UniProt and SwissLipids – MEYS Czech-Swiss project ELIXIR-IMPACT 8K0208 (2026–2028)
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