Conformational-Analysis-Guided Discovery of 2,3-Disubstituted Pyridine IDO1 Inhibitors.

Publication

Citation
Cherney EC, Zhang L, Guo W, Huang A, Williams D, Seitz S, Shan W, Zhu X, Gullo-Brown J, Maley D, Lin TA, Hunt JT, Huang C, Yang Z, D'Arienzo CJ, Discenza LN, Ranasinghe A, Grubb MF, Traeger SC, Li X, Johnston KA, Kopcho L, Fereshteh M, Foster KA, Stefanski K, Delpy D, Dhar G, Anandam A, Mahankali S, Padmanabhan S, Rajanna P, Murali V, Mariappan TT, Pattasseri S, Nimje RY, Hong Z, Kempson J, Rampulla R, Mathur A, Gupta A, Borzilleri R, Vite G, Balog A.: Conformational-Analysis-Guided Discovery of 2,3-Disubstituted Pyridine IDO1 Inhibitors. ACS Med Chem Lett, Volume 12 (7), 2021
Authors
Anandam A, Balog A., Borzilleri R, Cherney EC, D'Arienzo CJ, Delpy D, Dhar G, Discenza LN, Fereshteh M, Foster KA, Grubb MF, Gullo-Brown J, Guo W, Gupta A, Hong Z, Huang A, Huang C, Hunt JT, Johnston KA, Kempson J, Kopcho L, Li X, Lin TA, Mahankali S, Maley D, Mariappan TT, Mathur A, Murali V, Nimje RY, Padmanabhan S, Pattasseri S, Rajanna P, Rampulla R, Ranasinghe A, Seitz S, Shan W, Stefanski K, Traeger SC, Vite G, Williams D, Yang Z, Zhang L, Zhu X
Journal
ACS Med Chem Lett
Year
2021
PubMed
34267885
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Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

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  • MolMeDB interoperability with UniProt and SwissLipids – MEYS Czech-Swiss project ELIXIR-IMPACT 8K0208 (2026–2028)
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