- Citation
- Heightman TD, Berdini V, Braithwaite H, Buck IM, Cassidy M, Castro J, Courtin A, Day JEH, East C, Fazal L, Graham B, Griffiths-Jones CM, Lyons JF, Martins V, Muench S, Munck JM, Norton D, O'Reilly M, Palmer N, Pathuri P, Reader M, Rees DC, Rich SJ, Richardson C, Saini H, Thompson NT, Wallis NG, Walton H, Wilsher NE, Woolford AJ, Cooke M, Cousin D, Onions S, Shannon J, Watts J, Murray CW.: Fragment-Based Discovery of a Potent, Orally Bioavailable Inhibitor That Modulates the Phosphorylation and Catalytic Activity of ERK1/2. J Med Chem, Volume 61 (11), 2018
- Authors
- Berdini V, Braithwaite H, Buck IM, Cassidy M, Castro J, Cooke M, Courtin A, Cousin D, Day JEH, East C, Fazal L, Graham B, Griffiths-Jones CM, Heightman TD, Lyons JF, Martins V, Muench S, Munck JM, Murray CW., Norton D, O'Reilly M, Onions S, Palmer N, Pathuri P, Reader M, Rees DC, Rich SJ, Richardson C, Saini H, Shannon J, Thompson NT, Wallis NG, Walton H, Watts J, Wilsher NE, Woolford AJ
- Journal
- J Med Chem
- Year
- 2018
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