Citation

Marcoux D, Duan JJ, Shi Q, Cherney RJ, Srivastava AS, Cornelius L, Batt DG, Liu Q, Beaudoin-Bertrand M, Weigelt CA, Khandelwal P, Vishwakrishnan S, Selvakumar K, Karmakar A, Gupta AK, Basha M, Ramlingam S, Manjunath N, Vanteru S, Karmakar S, Maddala N, Vetrichelvan M, Gupta A, Rampulla RA, Mathur A, Yip S, Li P, Wu DR, Khan J, Ruzanov M, Sack JS, Wang J, Yarde M, Cvijic ME, Li S, Shuster DJ, Borowski V, Xie JH, McIntyre KW, Obermeier MT, Fura A, Stefanski K, Cornelius G, Hynes J, Tino JA, Macor JE, Salter-Cid L, Denton R, Zhao Q, Carter PH, Dhar TGM.: Rationally Designed, Conformationally Constrained Inverse Agonists of RORγt-Identification of a Potent, Selective Series with Biologic-Like in Vivo Efficacy. J Med Chem, Volume 62 (21), 2019

Authors

Basha M, Batt DG, Beaudoin-Bertrand M, Borowski V, Carter PH, Cherney RJ, Cornelius G, Cornelius L, Cvijic ME, Denton R, Dhar TGM., Duan JJ, Fura A, Gupta A, Gupta AK, Hynes J, Karmakar A, Karmakar S, Khan J, Khandelwal P, Li P, Li S, Liu Q, Macor JE, Maddala N, Manjunath N, Marcoux D, Mathur A, McIntyre KW, Obermeier MT, Ramlingam S, Rampulla RA, Ruzanov M, Sack JS, Salter-Cid L, Selvakumar K, Shi Q, Shuster DJ, Srivastava AS, Stefanski K, Tino JA, Vanteru S, Vetrichelvan M, Vishwakrishnan S, Wang J, Weigelt CA, Wu DR, Xie JH, Yarde M, Yip S, Zhao Q

Journal

J Med Chem

Year

2019

DOI

10.1021/acs.jmedchem.9b01369

PubMed

31638797

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