Discovery of BMS-986260, a Potent, Selective, and Orally Bioavailable TGFβR1 Inhibitor as an Immuno-oncology Agent.

Publication

Citation
Velaparthi U, Darne CP, Warrier J, Liu P, Rahaman H, Augustine-Rauch K, Parrish K, Yang Z, Swanson J, Brown J, Dhar G, Anandam A, Holenarsipur VK, Palanisamy K, Wautlet BS, Fereshteh MP, Lippy J, Tebben AJ, Sheriff S, Ruzanov M, Yan C, Gupta A, Gupta AK, Vetrichelvan M, Mathur A, Gelman M, Singh R, Kinsella T, Murtaza A, Fargnoli J, Vite G, Borzilleri RM.: Discovery of BMS-986260, a Potent, Selective, and Orally Bioavailable TGFβR1 Inhibitor as an Immuno-oncology Agent. ACS Med Chem Lett, Volume 11 (2), 2020
Authors
Anandam A, Augustine-Rauch K, Borzilleri RM., Brown J, Darne CP, Dhar G, Fargnoli J, Fereshteh MP, Gelman M, Gupta A, Gupta AK, Holenarsipur VK, Kinsella T, Lippy J, Liu P, Mathur A, Murtaza A, Palanisamy K, Parrish K, Rahaman H, Ruzanov M, Sheriff S, Singh R, Swanson J, Tebben AJ, Velaparthi U, Vetrichelvan M, Vite G, Warrier J, Wautlet BS, Yan C, Yang Z
Journal
ACS Med Chem Lett
Year
2020
PubMed
32071685
Machine-readable
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Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

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