Identification and optimisation of 7-azaindole PAK1 inhibitors with improved potency and kinase selectivity

Publication

Citation
McCoull, William; Edward J. Hennessy, Kevin Blades, Matthew R. Box, Claudio Chuaqui, James E. Dowling, Christopher D. Davies, Andrew D. Ferguson, Frederick W. Goldberg, Nicholas J. Howe, Paul D. Kemmitt, Gillian M. Lamont, Katrina Madden, Claire McWhirter, Jeffrey G. Varnes, Richard A. Ward, Jason D. Williams, Bin Yang: Identification and optimisation of 7-azaindole PAK1 inhibitors with improved potency and kinase selectivity. Med. Chem. Commun., 2014,5, 1533-1539, 10.1039/C4MD00280F
Authors
Andrew D. Ferguson, Bin Yang, Christopher D. Davies, Claire McWhirter, Claudio Chuaqui, Edward J. Hennessy, Frederick W. Goldberg, Gillian M. Lamont, James E. Dowling, Jason D. Williams, Jeffrey G. Varnes, Katrina Madden, Kevin Blades, Matthew R. Box, Nicholas J. Howe, Paul D. Kemmitt, Richard A. Ward, William McCoull
Journal
MedChemComm
Year
2014
Machine-readable
REST APIRDF
Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

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