Citation

Watterson SH, Liu Q, Beaudoin Bertrand M, Batt DG, Li L, Pattoli MA, Skala S, Cheng L, Obermeier MT, Moore R, Yang Z, Vickery R, Elzinga PA, Discenza L, D'Arienzo C, Gillooly KM, Taylor TL, Pulicicchio C, Zhang Y, Heimrich E, McIntyre KW, Ruan Q, Westhouse RA, Catlett IM, Zheng N, Chaudhry C, Dai J, Galella MA, Tebben AJ, Pokross M, Li J, Zhao R, Smith D, Rampulla R, Allentoff A, Wallace MA, Mathur A, Salter-Cid L, Macor JE, Carter PH, Fura A, Burke JR, Tino JA.: Discovery of Branebrutinib (BMS-986195): A Strategy for Identifying a Highly Potent and Selective Covalent Inhibitor Providing Rapid in Vivo Inactivation of Bruton's Tyrosine Kinase (BTK). J Med Chem, Volume 62 (7), 2019

Authors

Batt DG, Beaudoin Bertrand M, Cheng L, D'Arienzo C, Discenza L, Elzinga PA, Gillooly KM, Heimrich E, Li L, Liu Q, McIntyre KW, Moore R, Obermeier MT, Pattoli MA, Pulicicchio C, Skala S, Taylor TL, Vickery R, Watterson SH, Yang Z, Zhang Y, Allentoff A, Burke JR, Carter PH, Catlett IM, Chaudhry C, Dai J, Fura A, Galella MA, Li J, Macor JE, Mathur A, Pokross M, Rampulla R, Ruan Q, Salter-Cid L, Smith D, Tebben AJ, Tino JA., Wallace MA, Westhouse RA, Zhao R, Zheng N

Journal

J Med Chem

Year

2019

DOI

10.1021/acs.jmedchem.9b00167

PubMed

30893553

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