Inhibitors of human immunodeficiency virus type 1 (HIV-1) attachment. 12. Structure-activity relationships associated with 4-fluoro-6-azaindole derivatives leading to the identification of 1-(4-benzoylpiperazin-1-yl)-2-(4-fluoro-7-[1,2,3]triazol-1-yl-1h-pyrrolo[2,3-c]pyridin-3-yl)ethane-1,2-dione (BMS-585248).

Citation: Regueiro-Ren A, Xue QM, Swidorski JJ, Gong YF, Mathew M, Parker DD, Yang Z, Eggers B, D'Arienzo C, Sun Y, Malinowski J, Gao Q, Wu D, Langley DR, Colonno RJ, Chien C, Grasela DM, Zheng M, Lin PF, Meanwell NA, Kadow JF.: Inhibitors of human immunodeficiency virus type 1 (HIV-1) attachment. 12. Structure-activity relationships associated with 4-fluoro-6-azaindole derivatives leading to the identification of 1-(4-benzoylpiperazin-1-yl)-2-(4-fluoro-7-[1,2,3]triazol-1-yl-1h-pyrrolo[2,3-c]pyridin-3-yl)ethane-1,2-dione (BMS-585248). J Med Chem, Volume 56 (4), 2013
Authors: Colonno RJ, D'Arienzo C, Eggers B, Gao Q, Gong YF, Langley DR, Malinowski J, Mathew M, Parker DD, Regueiro-Ren A, Sun Y, Swidorski JJ, Wu D, Xue QM, Yang Z, Chien C, Grasela DM, Kadow JF., Lin PF, Meanwell NA, Zheng M
Journal: J Med Chem
Year: 2013
DOI: 10.1021/jm3016377
PubMed: 23360431
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