Discovery and optimization of a novel spiropyrrolidine inhibitor of β-secretase (BACE1) through fragment-based drug design.

Publication

Citation
Efremov IV, Vajdos FF, Borzilleri KA, Capetta S, Chen H, Dorff PH, Dutra JK, Goldstein SW, Mansour M, McColl A, Noell S, Oborski CE, O'Connell TN, O'Sullivan TJ, Pandit J, Wang H, Wei B, Withka JM.: Discovery and optimization of a novel spiropyrrolidine inhibitor of β-secretase (BACE1) through fragment-based drug design. J Med Chem, Volume 55 (21), 2012
Authors
Borzilleri KA, Capetta S, Chen H, Dorff PH, Dutra JK, Efremov IV, Goldstein SW, Mansour M, McColl A, Noell S, O'Connell TN, O'Sullivan TJ, Oborski CE, Pandit J, Vajdos FF, Wang H, Wei B, Withka JM.
Journal
J Med Chem
Year
2012
PubMed
22468999
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Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

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