- Citation
- Zehnder L, Bennett M, Meng J, Huang B, Ninkovic S, Wang F, Braganza J, Tatlock J, Jewell T, Zhou JZ, Burke B, Wang J, Maegley K, Mehta PP, Yin MJ, Gajiwala KS, Hickey MJ, Yamazaki S, Smith E, Kang P, Sistla A, Dovalsantos E, Gehring MR, Kania R, Wythes M, Kung PP.: Optimization of potent, selective, and orally bioavailable pyrrolodinopyrimidine-containing inhibitors of heat shock protein 90. Identification of development candidate 2-amino-4-{4-chloro-2-[2-(4-fluoro-1H-pyrazol-1-yl)ethoxy]-6-methylphenyl}-N-(2,2-difluoropropyl)-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxamide. J Med Chem, Volume 54 (9), 2011
- Authors
- Bennett M, Braganza J, Burke B, Dovalsantos E, Gajiwala KS, Gehring MR, Hickey MJ, Huang B, Jewell T, Kang P, Kania R, Kung PP., Maegley K, Mehta PP, Meng J, Ninkovic S, Sistla A, Smith E, Tatlock J, Wang F, Wang J, Wythes M, Yamazaki S, Yin MJ, Zehnder L, Zhou JZ
- Journal
- J Med Chem
- Year
- 2011
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