Citation

Terrett JA, Chen H, Shore DG, Villemure E, Larouche-Gauthier R, Déry M, Beaumier F, Constantineau-Forget L, Grand-Maître C, Lépissier L, Ciblat S, Sturino C, Chen Y, Hu B, Lu A, Wang Y, Cridland AP, Ward SI, Hackos DH, Reese RM, Shields SD, Chen J, Balestrini A, Riol-Blanco L, Lee WP, Liu J, Suto E, Wu X, Zhang J, Ly JQ, La H, Johnson K, Baumgardner M, Chou KJ, Rohou A, Rougé L, Safina BS, Magnuson S, Volgraf M.: Tetrahydrofuran-Based Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonists: Ligand-Based Discovery, Activity in a Rodent Asthma Model, and Mechanism-of-Action via Cryogenic Electron Microscopy. J Med Chem, Volume 64 (7), 2021

Authors

Balestrini A, Baumgardner M, Beaumier F, Chen H, Chen J, Chen Y, Chou KJ, Ciblat S, Constantineau-Forget L, Cridland AP, Déry M, Grand-Maître C, Hackos DH, Hu B, Johnson K, La H, Larouche-Gauthier R, Lee WP, Lépissier L, Liu J, Lu A, Ly JQ, Magnuson S, Reese RM, Riol-Blanco L, Rohou A, Rouge L, Safina BS, Shields SD, Shore DG, Sturino C, Suto E, Terrett JA, Villemure E, Volgraf M., Wang Y, Ward SI, Wu X, Zhang J

Journal

J Med Chem

Year

2021

DOI

10.1021/acs.jmedchem.0c02023

PubMed

33749283

Machine-readable

REST APIRDF