Citation

Chen H, Volgraf M, Do S, Kolesnikov A, Shore DG, Verma VA, Villemure E, Wang L, Chen Y, Hu B, Lu AJ, Wu G, Xu X, Yuen PW, Zhang Y, Erickson SD, Dahl M, Brotherton-Pleiss C, Tay S, Ly JQ, Murray LJ, Chen J, Amm D, Lange W, Hackos DH, Reese RM, Shields SD, Lyssikatos JP, Safina BS, Estrada AA.: Discovery of a Potent (4 R,5 S)-4-Fluoro-5-methylproline Sulfonamide Transient Receptor Potential Ankyrin 1 Antagonist and Its Methylene Phosphate Prodrug Guided by Molecular Modeling. J Med Chem, Volume 61 (8), 2018

Authors

Amm D, Brotherton-Pleiss C, Chen H, Chen J, Chen Y, Dahl M, Do S, Erickson SD, Estrada AA., Hackos DH, Hu B, Kolesnikov A, Lange W, Lu AJ, Ly JQ, Lyssikatos JP, Murray LJ, Reese RM, Safina BS, Shields SD, Shore DG, Tay S, Verma VA, Villemure E, Volgraf M, Wang L, Wu G, Xu X, Yuen PW, Zhang Y

Journal

J Med Chem

Year

2018

DOI

10.1021/acs.jmedchem.8b00117

PubMed

29590749

Machine-readable

REST APIRDF