Identification of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors with no evidence of CYP3A4 time-dependent inhibition and improved aqueous solubility.

Publication

Citation
Zak M, Liederer BM, Sampath D, Yuen PW, Bair KW, Baumeister T, Buckmelter AJ, Clodfelter KH, Cheng E, Crocker L, Fu B, Han B, Li G, Ho YC, Lin J, Liu X, Ly J, O'Brien T, Reynolds DJ, Skelton N, Smith CC, Tay S, Wang W, Wang Z, Xiao Y, Zhang L, Zhao G, Zheng X, Dragovich PS.: Identification of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors with no evidence of CYP3A4 time-dependent inhibition and improved aqueous solubility. Bioorg Med Chem Lett, Volume 25 (3), 2015
Authors
Bair KW, Baumeister T, Buckmelter AJ, Cheng E, Clodfelter KH, Crocker L, Dragovich PS., Fu B, Han B, Ho YC, Li G, Liederer BM, Lin J, Liu X, Ly J, O'Brien T, Reynolds DJ, Sampath D, Skelton N, Smith CC, Tay S, Wang W, Wang Z, Xiao Y, Yuen PW, Zak M, Zhang L, Zhao G, Zheng X
Journal
Bioorg Med Chem Lett
Year
2015
PubMed
25556090
Machine-readable
REST APIRDF
Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

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