Discovery of Acyl-sulfonamide Na<sub>v</sub>1.7 Inhibitors GDC-0276 and GDC-0310.

Publication

Citation
Safina BS, McKerrall SJ, Sun S, Chen CA, Chowdhury S, Jia Q, Li J, Zenova AY, Andrez JC, Bankar G, Bergeron P, Chang JH, Chang E, Chen J, Dean R, Decker SM, DiPasquale A, Focken T, Hemeon I, Khakh K, Kim A, Kwan R, Lindgren A, Lin S, Maher J, Mezeyova J, Misner D, Nelkenbrecher K, Pang J, Reese R, Shields SD, Sojo L, Sheng T, Verschoof H, Waldbrook M, Wilson MS, Xie Z, Young C, Zabka TS, Hackos DH, Ortwine DF, White AD, Johnson JP, Robinette CL, Dehnhardt CM, Cohen CJ, Sutherlin DP.: Discovery of Acyl-sulfonamide Na<sub>v</sub>1.7 Inhibitors GDC-0276 and GDC-0310. J Med Chem, Volume 64 (6), 2021
Authors
Andrez JC, Bankar G, Bergeron P, Chang E, Chang JH, Chen CA, Chen J, Chowdhury S, Cohen CJ, Dean R, Decker SM, Dehnhardt CM, DiPasquale A, Focken T, Hackos DH, Hemeon I, Jia Q, Johnson JP, Khakh K, Kim A, Kwan R, Li J, Lin S, Lindgren A, Maher J, McKerrall SJ, Mezeyova J, Misner D, Nelkenbrecher K, Ortwine DF, Pang J, Reese R, Robinette CL, Safina BS, Sheng T, Shields SD, Sojo L, Sun S, Sutherlin DP., Verschoof H, Waldbrook M, White AD, Wilson MS, Xie Z, Young C, Zabka TS, Zenova AY
Journal
J Med Chem
Year
2021
PubMed
33682420
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Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

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  • MolMeDB interoperability with UniProt and SwissLipids – MEYS Czech-Swiss project ELIXIR-IMPACT 8K0208 (2026–2028)
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