Challenges in the development of an M<sub>4</sub> PAM in vivo tool compound: The discovery of VU0467154 and unexpected DMPK profiles of close analogs.

Publication

Citation
Wood MR, Noetzel MJ, Poslusney MS, Melancon BJ, Tarr JC, Lamsal A, Chang S, Luscombe VB, Weiner RL, Cho HP, Bubser M, Jones CK, Niswender CM, Wood MW, Engers DW, Brandon NJ, Duggan ME, Conn PJ, Bridges TM, Lindsley CW.: Challenges in the development of an M<sub>4</sub> PAM in vivo tool compound: The discovery of VU0467154 and unexpected DMPK profiles of close analogs. Bioorg Med Chem Lett, Volume 27 (2), 2017
Authors
Brandon NJ, Bridges TM, Bubser M, Chang S, Cho HP, Conn PJ, Duggan ME, Engers DW, Jones CK, Lamsal A, Lindsley CW., Luscombe VB, Melancon BJ, Niswender CM, Noetzel MJ, Poslusney MS, Tarr JC, Weiner RL, Wood MR, Wood MW
Journal
Bioorg Med Chem Lett
Year
2017
PubMed
27939174
Machine-readable
REST APIRDF
Palacky University Olomouc

Palacky University Olomouc

Faculty of Science

Department of Physical Chemistry

tř. 17. listopadu 1192/12

771 46 Olomouc

Czech Republic

How to cite?

Juračka J., Šrejber M., Melíková M., Bazgier V., Berka K.: MolMeDB: Molecules on Membranes Database. Database, Volume 2019, 2019, baz078, https://doi.org/10.1093/database/baz078

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