{"data":{"id":841,"citation":"Pinard E, Alanine A, Alberati D, Bender M, Borroni E, Bourdeaux P, Brom V, Burner S, Fischer H, Hainzl D, Halm R, Hauser N, Jolidon S, Lengyel J, Marty HP, Meyer T, Moreau JL, Mory R, Narquizian R, Nettekoven M, Norcross RD, Puellmann B, Schmid P, Schmitt S, Stalder H, Wermuth R, Wettstein JG, Zimmerli D.: Selective GlyT1 inhibitors: discovery of [4-(3-fluoro-5-trifluoromethylpyridin-2-yl)piperazin-1-yl][5-methanesulfonyl-2-((S)-2,2,2-trifluoro-1-methylethoxy)phenyl]methanone (RG1678), a promising novel medicine to treat schizophrenia. J Med Chem, Volume 53 (12), 2010","title":"Selective GlyT1 inhibitors: discovery of [4-(3-fluoro-5-trifluoromethylpyridin-2-yl)piperazin-1-yl][5-methanesulfonyl-2-((S)-2,2,2-trifluoro-1-methylethoxy)phenyl]methanone (RG1678), a promising novel medicine to treat schizophrenia.","doi":"10.1021\/jm100210p","doi_url":"https:\/\/doi.org\/10.1021\/jm100210p","pmid":"20491477","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/20491477\/","year":2010,"journal":"J Med Chem","volume":"53","issue":"12","page":"4603-4614","authors":[{"first_name":"Alanine A","last_name":null,"full_name":null},{"first_name":"Alberati D","last_name":null,"full_name":null},{"first_name":"Bender M","last_name":null,"full_name":null},{"first_name":"Borroni E","last_name":null,"full_name":null},{"first_name":"Bourdeaux P","last_name":null,"full_name":null},{"first_name":"Brom V","last_name":null,"full_name":null},{"first_name":"Burner S","last_name":null,"full_name":null},{"first_name":"Fischer H","last_name":null,"full_name":null},{"first_name":"Hainzl D","last_name":null,"full_name":null},{"first_name":"Halm R","last_name":null,"full_name":null},{"first_name":"Hauser N","last_name":null,"full_name":null},{"first_name":"Jolidon S","last_name":null,"full_name":null},{"first_name":"Lengyel J","last_name":null,"full_name":null},{"first_name":"Marty HP","last_name":null,"full_name":null},{"first_name":"Meyer T","last_name":null,"full_name":null},{"first_name":"Moreau JL","last_name":null,"full_name":null},{"first_name":"Mory R","last_name":null,"full_name":null},{"first_name":"Narquizian R","last_name":null,"full_name":null},{"first_name":"Nettekoven M","last_name":null,"full_name":null},{"first_name":"Norcross RD","last_name":null,"full_name":null},{"first_name":"Pinard E","last_name":null,"full_name":null},{"first_name":"Puellmann B","last_name":null,"full_name":null},{"first_name":"Schmid P","last_name":null,"full_name":null},{"first_name":"Schmitt S","last_name":null,"full_name":null},{"first_name":"Stalder H","last_name":null,"full_name":null},{"first_name":"Wermuth R","last_name":null,"full_name":null},{"first_name":"Wettstein JG","last_name":null,"full_name":null},{"first_name":"Zimmerli D.","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/841","landing_page":"https:\/\/molmedb.upol.cz\/publication\/841","created_at":"2020-08-24T06:51:02.000000Z","updated_at":null}}