{"data":{"id":4802,"citation":"Brown A., Bagal S., Blackwell P., Blakemore D., Brown B., Bungay P., Corless M., Crawforth J., Fengas D., Fenwick D., Gray V., Kemp M., Klute W., Malet Sanz L., Miller D., Murata Y., Payne C., Skerratt S., Stevens E., Warmus J.: The discovery and optimization of benzimidazoles as selective NaV1.8 blockers for the treatment of pain. Bioorganic &amp; Medicinal Chemistry, Volume 27 (1), 2019","title":"The discovery and optimization of benzimidazoles as selective NaV1.8 blockers for the treatment of pain","doi":"10.1016\/j.bmc.2018.12.002","doi_url":"https:\/\/doi.org\/10.1016\/j.bmc.2018.12.002","pmid":null,"year":2019,"journal":"Bioorganic &amp; Medicinal Chemistry","volume":"27","issue":"1","page":null,"authors":[{"first_name":"Alan D.","last_name":"Brown","full_name":"Alan D. Brown"},{"first_name":"Sharan K.","last_name":"Bagal","full_name":"Sharan K. Bagal"},{"first_name":"Paul","last_name":"Blackwell","full_name":"Paul Blackwell"},{"first_name":"David C.","last_name":"Blakemore","full_name":"David C. Blakemore"},{"first_name":"Bruce","last_name":"Brown","full_name":"Bruce Brown"},{"first_name":"Peter J.","last_name":"Bungay","full_name":"Peter J. Bungay"},{"first_name":"Martin","last_name":"Corless","full_name":"Martin Corless"},{"first_name":"James","last_name":"Crawforth","full_name":"James Crawforth"},{"first_name":"David","last_name":"Fengas","full_name":"David Fengas"},{"first_name":"David R.","last_name":"Fenwick","full_name":"David R. Fenwick"},{"first_name":"Victoria","last_name":"Gray","full_name":"Victoria Gray"},{"first_name":"Mark","last_name":"Kemp","full_name":"Mark Kemp"},{"first_name":"Wolfgang","last_name":"Klute","full_name":"Wolfgang Klute"},{"first_name":"Laia","last_name":"Malet Sanz","full_name":"Laia Malet Sanz"},{"first_name":"Duncan","last_name":"Miller","full_name":"Duncan Miller"},{"first_name":"Yoshihisa","last_name":"Murata","full_name":"Yoshihisa Murata"},{"first_name":"C. Elizabeth","last_name":"Payne","full_name":"C. Elizabeth Payne"},{"first_name":"Sarah","last_name":"Skerratt","full_name":"Sarah Skerratt"},{"first_name":"Edward B.","last_name":"Stevens","full_name":"Edward B. Stevens"},{"first_name":"Joseph S.","last_name":"Warmus","full_name":"Joseph S. Warmus"}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/4802","landing_page":"https:\/\/molmedb.upol.cz\/publication\/4802","created_at":"2026-06-22T14:34:50.000000Z","updated_at":"2026-06-22T14:34:50.000000Z"}}