{"data":{"id":4615,"citation":"L\u00e9vesque JF, Bleasby K, Chefson A, Chen A, Dub\u00e9 D, Ducharme Y, Fournier PA, Gagn\u00e9 S, Gallant M, Grimm E, Hafey M, Han Y, Houle R, Lacombe P, Lalibert\u00e9 S, MacDonald D, Mackay B, Papp R, Tschirret-Guth R.: Impact of passive permeability and gut efflux transport on the oral bioavailability of novel series of piperidine-based renin inhibitors in rodents. Bioorg Med Chem Lett, Volume 21 (18), 2011","title":"Impact of passive permeability and gut efflux transport on the oral bioavailability of novel series of piperidine-based renin inhibitors in rodents.","doi":"10.1016\/j.bmcl.2011.06.095","doi_url":"https:\/\/doi.org\/10.1016\/j.bmcl.2011.06.095","pmid":"21784634","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/21784634\/","year":2011,"journal":"Bioorg Med Chem Lett","volume":"21","issue":"18","page":"5547-5551","authors":[{"first_name":"Bleasby K","last_name":null,"full_name":null},{"first_name":"Chefson A","last_name":null,"full_name":null},{"first_name":"Chen A","last_name":null,"full_name":null},{"first_name":"Dub\u00e9 D","last_name":null,"full_name":null},{"first_name":"Ducharme Y","last_name":null,"full_name":null},{"first_name":"Fournier PA","last_name":null,"full_name":null},{"first_name":"Gagn\u00e9 S","last_name":null,"full_name":null},{"first_name":"Gallant M","last_name":null,"full_name":null},{"first_name":"Grimm E","last_name":null,"full_name":null},{"first_name":"Hafey M","last_name":null,"full_name":null},{"first_name":"Han Y","last_name":null,"full_name":null},{"first_name":"Houle R","last_name":null,"full_name":null},{"first_name":"Lacombe P","last_name":null,"full_name":null},{"first_name":"Lalibert\u00e9 S","last_name":null,"full_name":null},{"first_name":"L\u00e9vesque JF","last_name":null,"full_name":null},{"first_name":"MacDonald D","last_name":null,"full_name":null},{"first_name":"Mackay B","last_name":null,"full_name":null},{"first_name":"Papp R","last_name":null,"full_name":null},{"first_name":"Tschirret-Guth R.","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/4615","landing_page":"https:\/\/molmedb.upol.cz\/publication\/4615","created_at":"2024-08-12T07:48:27.000000Z","updated_at":null}}