{"data":{"id":4239,"citation":"Liu YA, Jin Q, Zou Y, Ding Q, Yan S, Wang Z, Hao X, Nguyen B, Zhang X, Pan J, Mo T, Jacobsen K, Lam T, Wu TY, Petrassi HM, Bursulaya B, DiDonato M, Gordon WP, Liu B, Baaten J, Hill R, Nguyen-Tran V, Qiu M, Zhang YQ, Kamireddy A, Espinola S, Deaton L, Ha S, Harb G, Jia Y, Li J, Shen W, Schumacher AM, Colman K, Glynne R, Pan S, McNamara P, Laffitte B, Meeusen S, Molteni V, Loren J.: Selective DYRK1A Inhibitor for the Treatment of Type 1 Diabetes: Discovery of 6-Azaindole Derivative GNF2133. J Med Chem, Volume 63 (6), 2020","title":"Selective DYRK1A Inhibitor for the Treatment of Type 1 Diabetes: Discovery of 6-Azaindole Derivative GNF2133.","doi":"10.1021\/acs.jmedchem.9b01624","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.9b01624","pmid":"32077280","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/32077280\/","year":2020,"journal":"J Med Chem","volume":"63","issue":"6","page":"2958-2973","authors":[{"first_name":"Ding Q","last_name":null,"full_name":null},{"first_name":"Hao X","last_name":null,"full_name":null},{"first_name":"Jin Q","last_name":null,"full_name":null},{"first_name":"Liu YA","last_name":null,"full_name":null},{"first_name":"Wang Z","last_name":null,"full_name":null},{"first_name":"Yan S","last_name":null,"full_name":null},{"first_name":"Zou Y","last_name":null,"full_name":null},{"first_name":"Baaten J","last_name":null,"full_name":null},{"first_name":"Bursulaya B","last_name":null,"full_name":null},{"first_name":"Colman K","last_name":null,"full_name":null},{"first_name":"Deaton L","last_name":null,"full_name":null},{"first_name":"DiDonato M","last_name":null,"full_name":null},{"first_name":"Espinola S","last_name":null,"full_name":null},{"first_name":"Glynne R","last_name":null,"full_name":null},{"first_name":"Gordon WP","last_name":null,"full_name":null},{"first_name":"Ha S","last_name":null,"full_name":null},{"first_name":"Harb G","last_name":null,"full_name":null},{"first_name":"Hill R","last_name":null,"full_name":null},{"first_name":"Jacobsen K","last_name":null,"full_name":null},{"first_name":"Jia Y","last_name":null,"full_name":null},{"first_name":"Kamireddy A","last_name":null,"full_name":null},{"first_name":"Laffitte B","last_name":null,"full_name":null},{"first_name":"Lam T","last_name":null,"full_name":null},{"first_name":"Li J","last_name":null,"full_name":null},{"first_name":"Liu B","last_name":null,"full_name":null},{"first_name":"Loren J.","last_name":null,"full_name":null},{"first_name":"McNamara P","last_name":null,"full_name":null},{"first_name":"Meeusen S","last_name":null,"full_name":null},{"first_name":"Mo T","last_name":null,"full_name":null},{"first_name":"Molteni V","last_name":null,"full_name":null},{"first_name":"Nguyen B","last_name":null,"full_name":null},{"first_name":"Nguyen-Tran V","last_name":null,"full_name":null},{"first_name":"Pan J","last_name":null,"full_name":null},{"first_name":"Pan S","last_name":null,"full_name":null},{"first_name":"Petrassi HM","last_name":null,"full_name":null},{"first_name":"Qiu M","last_name":null,"full_name":null},{"first_name":"Schumacher AM","last_name":null,"full_name":null},{"first_name":"Shen W","last_name":null,"full_name":null},{"first_name":"Wu TY","last_name":null,"full_name":null},{"first_name":"Zhang X","last_name":null,"full_name":null},{"first_name":"Zhang YQ","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/4239","landing_page":"https:\/\/molmedb.upol.cz\/publication\/4239","created_at":"2024-05-24T08:49:33.000000Z","updated_at":null}}