{"data":{"id":4203,"citation":"Klein VG, Bond AG, Craigon C, Lokey RS, Ciulli A.: Amide-to-Ester Substitution as a Strategy for Optimizing PROTAC Permeability and Cellular Activity. J Med Chem, Volume 64 (24), 2021","title":"Amide-to-Ester Substitution as a Strategy for Optimizing PROTAC Permeability and Cellular Activity.","doi":"10.1021\/acs.jmedchem.1c01496","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.1c01496","pmid":"34881891","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/34881891\/","year":2021,"journal":"J Med Chem","volume":"64","issue":"24","page":"18082-18101","authors":[{"first_name":"Bond AG","last_name":null,"full_name":null},{"first_name":"Ciulli A.","last_name":null,"full_name":null},{"first_name":"Craigon C","last_name":null,"full_name":null},{"first_name":"Klein VG","last_name":null,"full_name":null},{"first_name":"Lokey RS","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/4203","landing_page":"https:\/\/molmedb.upol.cz\/publication\/4203","created_at":"2024-05-24T08:49:16.000000Z","updated_at":null}}