{"data":{"id":4191,"citation":"Naidu BN, Patel M, McAuliffe B, Ding B, Cianci C, Simmermacher J, Jenkins S, Parker DD, Sivaprakasam P, Khan JA, Kish K, Lewis H, Hanumegowda U, Krystal M, Meanwell NA, Kadow JF.: Design, Synthesis, and Preclinical Profiling of GSK3739936 (BMS-986180), an Allosteric Inhibitor of HIV-1 Integrase with Broad-Spectrum Activity toward 124\/125 Polymorphs. J Med Chem, Volume 65 (6), 2022","title":"Design, Synthesis, and Preclinical Profiling of GSK3739936 (BMS-986180), an Allosteric Inhibitor of HIV-1 Integrase with Broad-Spectrum Activity toward 124\/125 Polymorphs.","doi":"10.1021\/acs.jmedchem.1c02169","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.1c02169","pmid":"35235334","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/35235334\/","year":2022,"journal":"J Med Chem","volume":"65","issue":"6","page":"4949-4971","authors":[{"first_name":"Cianci C","last_name":null,"full_name":null},{"first_name":"Ding B","last_name":null,"full_name":null},{"first_name":"Hanumegowda U","last_name":null,"full_name":null},{"first_name":"Jenkins S","last_name":null,"full_name":null},{"first_name":"Kadow JF.","last_name":null,"full_name":null},{"first_name":"Khan JA","last_name":null,"full_name":null},{"first_name":"Kish K","last_name":null,"full_name":null},{"first_name":"Krystal M","last_name":null,"full_name":null},{"first_name":"Lewis H","last_name":null,"full_name":null},{"first_name":"McAuliffe B","last_name":null,"full_name":null},{"first_name":"Meanwell NA","last_name":null,"full_name":null},{"first_name":"Naidu BN","last_name":null,"full_name":null},{"first_name":"Parker DD","last_name":null,"full_name":null},{"first_name":"Patel M","last_name":null,"full_name":null},{"first_name":"Simmermacher J","last_name":null,"full_name":null},{"first_name":"Sivaprakasam P","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/4191","landing_page":"https:\/\/molmedb.upol.cz\/publication\/4191","created_at":"2024-05-24T08:49:10.000000Z","updated_at":null}}