{"data":{"id":4188,"citation":"Velcicky J, Wilcken R, Cotesta S, Janser P, Schlapbach A, Wagner T, Piechon P, Villard F, Bouhelal R, Piller F, Harlfinger S, Stringer R, Fehlmann D, Kaupmann K, Littlewood-Evans A, Haffke M, Gommermann N.: Discovery and Optimization of Novel SUCNR1 Inhibitors: Design of Zwitterionic Derivatives with a Salt Bridge for the Improvement of Oral Exposure. J Med Chem, Volume 63 (17), 2020","title":"Discovery and Optimization of Novel SUCNR1 Inhibitors: Design of Zwitterionic Derivatives with a Salt Bridge for the Improvement of Oral Exposure.","doi":"10.1021\/acs.jmedchem.0c01020","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.0c01020","pmid":"32856916","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/32856916\/","year":2020,"journal":"J Med Chem","volume":"63","issue":"17","page":"9856-9875","authors":[{"first_name":"Bouhelal R","last_name":null,"full_name":null},{"first_name":"Cotesta S","last_name":null,"full_name":null},{"first_name":"Fehlmann D","last_name":null,"full_name":null},{"first_name":"Gommermann N.","last_name":null,"full_name":null},{"first_name":"Haffke M","last_name":null,"full_name":null},{"first_name":"Harlfinger S","last_name":null,"full_name":null},{"first_name":"Janser P","last_name":null,"full_name":null},{"first_name":"Kaupmann K","last_name":null,"full_name":null},{"first_name":"Littlewood-Evans A","last_name":null,"full_name":null},{"first_name":"Piechon P","last_name":null,"full_name":null},{"first_name":"Piller F","last_name":null,"full_name":null},{"first_name":"Schlapbach A","last_name":null,"full_name":null},{"first_name":"Stringer R","last_name":null,"full_name":null},{"first_name":"Velcicky J","last_name":null,"full_name":null},{"first_name":"Villard F","last_name":null,"full_name":null},{"first_name":"Wagner T","last_name":null,"full_name":null},{"first_name":"Wilcken R","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/4188","landing_page":"https:\/\/molmedb.upol.cz\/publication\/4188","created_at":"2024-05-24T08:49:09.000000Z","updated_at":null}}