{"data":{"id":4139,"citation":"Milite C, Feoli A, Horton JR, Rescigno D, Cipriano A, Pisapia V, Viviano M, Pepe G, Amendola G, Novellino E, Cosconati S, Cheng X, Castellano S, Sbardella G.: Discovery of a Novel Chemotype of Histone Lysine Methyltransferase EHMT1\/2 (GLP\/G9a) Inhibitors: Rational Design, Synthesis, Biological Evaluation, and Co-crystal Structure. J Med Chem, Volume 62 (5), 2019","title":"Discovery of a Novel Chemotype of Histone Lysine Methyltransferase EHMT1\/2 (GLP\/G9a) Inhibitors: Rational Design, Synthesis, Biological Evaluation, and Co-crystal Structure.","doi":"10.1021\/acs.jmedchem.8b02008","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.8b02008","pmid":"30753076","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/30753076\/","year":2019,"journal":"J Med Chem","volume":"62","issue":"5","page":"2666-2689","authors":[{"first_name":"Amendola G","last_name":null,"full_name":null},{"first_name":"Castellano S","last_name":null,"full_name":null},{"first_name":"Cheng X","last_name":null,"full_name":null},{"first_name":"Cipriano A","last_name":null,"full_name":null},{"first_name":"Cosconati S","last_name":null,"full_name":null},{"first_name":"Feoli A","last_name":null,"full_name":null},{"first_name":"Horton JR","last_name":null,"full_name":null},{"first_name":"Milite C","last_name":null,"full_name":null},{"first_name":"Novellino E","last_name":null,"full_name":null},{"first_name":"Pepe G","last_name":null,"full_name":null},{"first_name":"Pisapia V","last_name":null,"full_name":null},{"first_name":"Rescigno D","last_name":null,"full_name":null},{"first_name":"Sbardella G.","last_name":null,"full_name":null},{"first_name":"Viviano M","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/4139","landing_page":"https:\/\/molmedb.upol.cz\/publication\/4139","created_at":"2024-05-23T10:43:11.000000Z","updated_at":null}}