{"data":{"id":4134,"citation":"Wilson C, Ray P, Zuccotto F, Hernandez J, Aggarwal A, Mackenzie C, Caldwell N, Taylor M, Huggett M, Mathieson M, Murugesan D, Smith A, Davis S, Cocco M, Parai MK, Acharya A, Tamaki F, Scullion P, Epemolu O, Riley J, Stojanovski L, Lopez-Rom\u00e1n EM, Torres-G\u00f3mez PA, Toledo AM, Guijarro-Lopez L, Camino I, Engelhart CA, Schnappinger D, Massoudi LM, Lenaerts A, Robertson GT, Walpole C, Matthews D, Floyd D, Sacchettini JC, Read KD, Encinas L, Bates RH, Green SR, Wyatt PG.: Optimization of TAM16, a Benzofuran That Inhibits the Thioesterase Activity of Pks13; Evaluation toward a Preclinical Candidate for a Novel Antituberculosis Clinical Target. J Med Chem, Volume 65 (1), 2022","title":"Optimization of TAM16, a Benzofuran That Inhibits the Thioesterase Activity of Pks13; Evaluation toward a Preclinical Candidate for a Novel Antituberculosis Clinical Target.","doi":"10.1021\/acs.jmedchem.1c01586","doi_url":"https:\/\/doi.org\/10.1021\/acs.jmedchem.1c01586","pmid":"34910486","pmid_url":"https:\/\/pubmed.ncbi.nlm.nih.gov\/34910486\/","year":2022,"journal":"J Med Chem","volume":"65","issue":"1","page":"409-423","authors":[{"first_name":"Acharya A","last_name":null,"full_name":null},{"first_name":"Aggarwal A","last_name":null,"full_name":null},{"first_name":"Bates RH","last_name":null,"full_name":null},{"first_name":"Caldwell N","last_name":null,"full_name":null},{"first_name":"Camino I","last_name":null,"full_name":null},{"first_name":"Cocco M","last_name":null,"full_name":null},{"first_name":"Davis S","last_name":null,"full_name":null},{"first_name":"Encinas L","last_name":null,"full_name":null},{"first_name":"Engelhart CA","last_name":null,"full_name":null},{"first_name":"Epemolu O","last_name":null,"full_name":null},{"first_name":"Floyd D","last_name":null,"full_name":null},{"first_name":"Green SR","last_name":null,"full_name":null},{"first_name":"Guijarro-Lopez L","last_name":null,"full_name":null},{"first_name":"Hernandez J","last_name":null,"full_name":null},{"first_name":"Huggett M","last_name":null,"full_name":null},{"first_name":"Lenaerts A","last_name":null,"full_name":null},{"first_name":"L\u00f3pez-Rom\u00e1n EM","last_name":null,"full_name":null},{"first_name":"Mackenzie C","last_name":null,"full_name":null},{"first_name":"Massoudi LM","last_name":null,"full_name":null},{"first_name":"Mathieson M","last_name":null,"full_name":null},{"first_name":"Matthews D","last_name":null,"full_name":null},{"first_name":"Murugesan D","last_name":null,"full_name":null},{"first_name":"Parai MK","last_name":null,"full_name":null},{"first_name":"Ray P","last_name":null,"full_name":null},{"first_name":"Read KD","last_name":null,"full_name":null},{"first_name":"Riley J","last_name":null,"full_name":null},{"first_name":"Robertson GT","last_name":null,"full_name":null},{"first_name":"Sacchettini JC","last_name":null,"full_name":null},{"first_name":"Schnappinger D","last_name":null,"full_name":null},{"first_name":"Scullion P","last_name":null,"full_name":null},{"first_name":"Smith A","last_name":null,"full_name":null},{"first_name":"Stojanovski L","last_name":null,"full_name":null},{"first_name":"Tamaki F","last_name":null,"full_name":null},{"first_name":"Taylor M","last_name":null,"full_name":null},{"first_name":"Toledo AM","last_name":null,"full_name":null},{"first_name":"Torres-G\u00f3mez PA","last_name":null,"full_name":null},{"first_name":"Walpole C","last_name":null,"full_name":null},{"first_name":"Wilson C","last_name":null,"full_name":null},{"first_name":"Wyatt PG.","last_name":null,"full_name":null},{"first_name":"Zuccotto F","last_name":null,"full_name":null}],"url":"https:\/\/molmedb.upol.cz\/api\/v1\/publications\/4134","landing_page":"https:\/\/molmedb.upol.cz\/publication\/4134","created_at":"2024-05-23T10:43:09.000000Z","updated_at":null}}